Therapeutic Compounds and Approaches
Use of a Novel 5′‐Regioselective Phosphitylating Reagent for One‐Pot Synthesis of Nucleoside 5′‐Triphosphates from Unprotected Nucleosides
Julianne Caton‐Williams, Rudiona Hoxhaj, Bilal Fiaz, Zhen Huang
Published online: March 2013
Julianne Caton‐Williams, Rudiona Hoxhaj, Bilal Fiaz, Zhen Huang
Published online: March 2013
Synthesis of a North‐Methanocarba‐Thymidine (N‐MCT) Analog
Andrew Thompson, Victor E. Marquez
Published online: December 2012
Andrew Thompson, Victor E. Marquez
Published online: December 2012
Binding to the DNA Minor Groove by Heterocyclic Dications: From AT‐Specific Monomers to GC Recognition with Dimers
Rupesh Nanjunda, W. David Wilson
Published online: December 2012
Rupesh Nanjunda, W. David Wilson
Published online: December 2012
Preparation of Azido Containing Oligonucleotides Through Diazo Transfer Reaction
Rémy Lartia, Laureen Bonnat, Pierre Murat, Eric Defrancq
Published online: September 2012
Rémy Lartia, Laureen Bonnat, Pierre Murat, Eric Defrancq
Published online: September 2012
Sequence, Stability, and Structure of G‐Quadruplexes and Their Interactions with Drugs
Yuwei Chen, Danzhou Yang, Danzhou Yang, Danzhou Yang, Danzhou Yang
Published online: September 2012
Yuwei Chen, Danzhou Yang, Danzhou Yang, Danzhou Yang, Danzhou Yang
Published online: September 2012
Two‐Step, One‐Pot Synthesis of Inosine, Guanosine, and 2′‐Deoxyguanosine O6‐Ethers via Intermediate O6‐(Benzotriazol‐1‐yl) Derivatives
Hari Prasad Kokatla, Mahesh K. Lakshman
Published online: June 2012
Hari Prasad Kokatla, Mahesh K. Lakshman
Published online: June 2012
Oligodeoxynucleotide Containing S‐Functionalized 2′‐Deoxy‐6‐Thioguanosine: Facile Tools for Base‐Selective and Site‐Specific Internal Modification of RNA
Shigeki Sasaki, Kazumitsu Onizuka, Yosuke Taniguchi
Published online: March 2012
Shigeki Sasaki, Kazumitsu Onizuka, Yosuke Taniguchi
Published online: March 2012
Synthesis of Dumbbell‐Shaped Cyclic RNAs for RNA Interference
Naoko Abe, Hiroshi Abe, Yoshihiro Ito
Published online: March 2012
Naoko Abe, Hiroshi Abe, Yoshihiro Ito
Published online: March 2012
Synthesis of Entecavir and Its Novel Class of Analogs
Ravindra K. Rawal, Uma Sharan Singh, Srinivas Gadthula, Chung K. Chu
Published online: December 2011
Ravindra K. Rawal, Uma Sharan Singh, Srinivas Gadthula, Chung K. Chu
Published online: December 2011
A Status Update of Modified Oligonucleotides for Chemotherapeutics Applications
Yogesh S. Sanghvi
Published online: September 2011
Yogesh S. Sanghvi
Published online: September 2011
RNA Aptamers and Spiegelmers: Synthesis, Purification, and Post‐Synthetic PEG Conjugation
Stefanie Hoffmann, Johannes Hoos, Sven Klussmann, Stefan Vonhoff
Published online: September 2011
Stefanie Hoffmann, Johannes Hoos, Sven Klussmann, Stefan Vonhoff
Published online: September 2011
Synthesis of 2′,4′‐Bridged Nucleosides Using a New Orthogonally Protected Sugar Synthon: 5‐O‐(tert‐Butyldiphenylsilyl)‐4‐C‐Hydroxymethyl‐1,2‐O‐Isopropylidene‐3‐O‐Napthyl‐α‐d‐Allofuranose
Punit P. Seth, Thazha P. Prakash
Published online: March 2011
Punit P. Seth, Thazha P. Prakash
Published online: March 2011
Time‐Dependent Thermocontrol of the Hydrophilic and Lipophilic Properties of DNA Oligonucleotide Prodrugs
Cristina Ausín, Andrzej Grajkowski, Jacek Cieślak, Alexei Gapeev, Serge L. Beaucage
Published online: December 2010
Cristina Ausín, Andrzej Grajkowski, Jacek Cieślak, Alexei Gapeev, Serge L. Beaucage
Published online: December 2010
Synthesis of Peptidomimetic Conjugates of Cyclic Nucleoside Phosphonates
Michaela Serpi, Ivan S. Krylov, Valeria M. Zakharova, Charles E. McKenna
Published online: December 2010
Michaela Serpi, Ivan S. Krylov, Valeria M. Zakharova, Charles E. McKenna
Published online: December 2010
In Vitro Selection of RNA Aptamers to a Small Molecule Target
Vlad Codrea, Michelle Hayner, Bradley Hall, Sulay Jhaveri, Andrew Ellington
Published online: March 2010
Vlad Codrea, Michelle Hayner, Bradley Hall, Sulay Jhaveri, Andrew Ellington
Published online: March 2010
Nucleoside Modification with Boron Clusters and Their Metal Complexes
Blazej A. Wojtczak, Agnieszka B. Olejniczak, Zbigniew J. Lesnikowski
Published online: September 2009
Blazej A. Wojtczak, Agnieszka B. Olejniczak, Zbigniew J. Lesnikowski
Published online: September 2009
Solid‐Supported Reagents for Synthesis of Nucleoside Monothiophosphates, Dithiodiphosphates, and Trithiotriphosphates
Yousef Ahmadibeni, Keykavous Parang
Published online: March 2009
Yousef Ahmadibeni, Keykavous Parang
Published online: March 2009
A Universal and Recyclable Solid Support for Oligonucleotide Synthesis
François Morvan, Albert Meyer, Jean‐Jacques Vasseur
Published online: September 2007
François Morvan, Albert Meyer, Jean‐Jacques Vasseur
Published online: September 2007
Solution‐Phase Synthesis of Di‐ and Trinucleotides Using Polymer‐Supported Reagents
François Morvan, Jean‐Jacques Vasseur
Published online: October 2006
François Morvan, Jean‐Jacques Vasseur
Published online: October 2006



